Publications (since July 2013)
Book chapters
Book chapters
Scientific articles
87. D. Moita, T.G. Maia, M. Duarte, C.M. Andrade, I.S. Albuquerque, A. Dwivedi, J.C. Silva, L. González-Céron, C.J. Janse, A.M. Mendes, M. Prudêncio (2022) “A genetically modified Plasmodium berghei parasite as a surrogate for whole-sporozoite vaccination against P. vivax malaria”, NPJ Vaccines, 7, 163, 1-9
86. B. Franke-Fayard, C. Marin-Mogollon, F.J.A. Geurten, S. Chevalley-Maurel, J. Ramesar, H. Kroeze, E Baalbergen, E. Wessels, L. Baron, V. Soulard, T. Martinson, M. Aleshnick, A.T.G. Huijs, A.K. Subudhi, Y. Miyazaki, A.S. Othman, S. K. Kolli, O.A.C. Lamers, M. Roques, R.R. Stanway, S.C. Murphy, L. Foquet, D. Moita, A.M. Mendes, M. Prudêncio, K.J. Dechering, V.T. Heussler, A. Pain., B.K. Wilder, M. Roestenberg, C.J. Janse (2022) “Creation and preclinical 1 evaluation of genetically attenuated malaria parasites arresting growth late in the liver”, NPJ Vaccines, 7, 139, 1-17
85. A.J. Alves, N.G. Alves, I. Bártolo, D. Fontinha, S. Caetano, M. Prudêncio, N.Taveira, T.M. Pinho e Melo (2022) “Unveiling a family of spiro‐beta‐lactams with anti-HIV and anti-plasmodial activity via phosphine-catalyzed [3+2] annulation of 6-alkylidene-penicillanates and allenoates”, Front. Chem., 10, 1017250
84. H. Nunes-Cabaço, D. Moita, M. Prudêncio (2022) "Five decades of clinical assessment of whole-sporozoite malaria vaccines", Front. Immunol., 13, 977472
83. I. Bouzón-Arnáiz; Y. Avalos-Padilla; A. Biosca; O. Caño-Prades; L. Román-Álamo; J. Valle; D. Andreu; D. Moita; M. Prudêncio; E.M. Arce; D. Muñoz-Torrero; X. Fernàndez-Busquets (2022) “The protein aggregation inhibitor YAT2150 has potent antimalarial activity in Plasmodium falciparum in vitro cultures", BMC Biology, 20, 197, 1-27
82. Y. Le Gal, A. Filatre-Furcate, D. Lorcy, O. Jeannin, T. Roisnel, V. Dorcet, D. Fontinha, D. Francisco, M. Prudêncio, M. Martins, C. Soeiro, S.A. Sousa, J.H. Leitão, T.S. Morais, I. Bártolo, N. Taveira, J.F. Guerreiro, F. Marques (2022) “Broad Spectrum Functional Activity of Structurally Related Monoanionic Au(III) Bis(Dithiolene) Complexes”, Int. J. Mol. Sci., 23, 7146
81. C.S. Pereira, H.C. Quadros, S.Y. Aboagye, D. Fontinha, S. D’Alessandro, M.E. Byrne, M. Gendrot, I. Fonta, J. Mosnier, D. Rodrigo, M. Moreira, N. Basilico, D.L. Williams, M. Prudêncio, B. Pradines, M. Navarro (2022) "Hybrid of amodiaquine and primaquine linked by gold(I) is a multistage antimalarial agent by targeting heme detoxification and thiol redox homeostasis", Pharmaceutics, 14, 1251
80. A. Khandelwal, F. Arez, P.M. Alves, L. Badolo, C. Brito, C. Fischli, D. Fontinha, C. Oeuvray, M. Prudêncio, M. Rottmann, J. Wilkins, Ö. Yalkinoglu, W.M. Bagchus, T. Spangenberg (2022) “Translation of liver stage activity of M5717, a Plasmodium Elongation Factor 2 inhibitor - from bench to bedside”, Malaria J., 21, 151
79. H. Nunes-Cabaço, D. Moita, C. Rôla, A.M. Mendes, M. Prudêncio (2022) “Impact of dietary protein restriction on the immunogenicity and efficacy of whole-sporozoite malaria vaccination”, Front. Immunol., 13, 869757
78. E.A. Lopes, R. Mestre, D. Fontinha, J. Legac, J.V. Pei, M. Sanches-Vaz, M. Mori, A.M. Lehane, P.J. Rosenthal, M. Prudêncio, M.M.M. Santos (2022) “Discovery of spirooxadiazoline oxindoles with dual-stage antimalarial activity”, Eur. J. Med. Chem., 236, 114324
77. D. Jublot, P. Cavaillès, S. Kamche, D. Francisco, D. Fontinha, M. Prudêncio, J.-F. Guichou, G. Labesse, D. Sereno, C. Loeuillet (2022) "A Histone deacetylase (HDAC) inhibitor with pleiotropic in vitro anti-Toxoplasma and Plasmodial activities controls acute and chronic toxoplasma infection in mice", Int. J. Mol. Sci., 23, 3254
76. D. Fontinha*, F. Arez*, I.R. Gal, G. Nogueira, D. Moita, T.H.H. Baeurle, C. Brito, T. Spangenberg**, P.M. Alves**, M. Prudêncio** (2022) "Pre-erythrocytic activity of M5717 in monotherapy and combination in preclinical Plasmodium infection models", ACS Inf. Dis., 8, 721-727. *Equally contributing authors; **Corresponding authors.
75. A.F. Chora, M.M. Mota, M. Prudêncio (2022) "The reciprocal influence of the liver and blood stages of the malaria parasite's life cycle", Int. J. Parasitol., 52, 711-715
74. S. Portugal, A. Rodriguez, M. Prudêncio (2022) “Maria M. Mota: Bringing Plasmodium Liver Infection to the Centre Stage of Malaria Research”, Front. Cell. Infect. Microbiol., 12, 851484
73. L. Singh, D. Fontinha, D. Francisco, M. Prudêncio, K. Singh (2022) “Synthesis and Antiplasmodial Activity of Regioisomers and Epimers of Second-Generation Dual Acting Ivermectin Hybrids“, Sci. Rep., 12,564
72. C. Upadhyay, N. Sharma, S. Kumar, P.P. Sharma, D. Fontinha, B.S. Chhikara, B. Mukherjee, D. Kumar, M. Prudêncio, A.P. Singh, Poonam (2022) “Synthesis of the new analogs of morpholine and their antiplasmodial evaluation against the human malaria parasite Plasmodium falciparum", New. J. Chem., 46, 250
71. A.T. Silva, I.S. Oliveira, J. Gomes, L. Aguiar, D. Fontinha, D. Duarte, F. Nogueira, M. Prudêncio, E.F. Marques, C. Teixeira, R. Ferraz, P. Gomes (2021) “Drug-derived surface-active ionic liquids: a cost-effective way to expressively increase blood-stage antimalarial activity of primaquine“, ChemMedChem, e202100650
70. H.C. Quadros, A. Çapcı, L. Herrmann, S. D’Alessandro, D. Fontinha, R. Azevedo, W. Villarreal, N. Basilico, M. Prudêncio, S.B. Tsogoeva, D.R.M. Moreira (2021) “Studies of Potency and Efficacy of an Optimized Dihydroartemisinin-Quinoline Hybrid against Multiple Stages of the Plasmodium Life Cycle”, Pharmaceuticals, 14, 1129
69. T. Araki*, J. Lin*, M. Prudêncio*, D.A. Cunningham*, T. Annoura* (2021), “Editorial Malaria Targeting Toolkit: Host-Parasite Interactions” Front. Cell. Infect. Microbiol., 11, 79549. *Corresponding authors
68. A. Temporão*, M. Sanches-Vaz*, R. Luís, H. Nunes-Cabaço, T.K. Smith, M. Prudêncio**, L. Figueiredo** (2021) "Excreted Trypanosoma brucei proteins inhibit Plasmodium hepatic infection", PLoS Negl. Trop. Dis., October 29. * Equally contributing authors; **Corresponding authors. Recommended by Faculty Opinions.
67. M. Marinović, G. Poje, I. Perković, D. Fontinha, M. Prudêncio, J. Held, L.P. Carvalho, T. Tandarić, R. Vianello, Z. Rajić (2021), “Further investigation of harmicines as novel antiplasmodial agents: Synthesis,structure-activity relationship and insight into the mechanism of action”, Eur. J. Med. Chem., 224, 113687
66. C.S. Pereira, H.C. Quadros, D.R.M. Moreira, W. Castro, Silva R.I.S.D.S., M.B.P. Soares, D. Fontinha, M. Prudêncio, V. Schmitz, H.F. Santos, M. Gendrot, I. Fonta, J. Mosnier, B. Pradines, M.Navarro (2021), “A Novel Hybrid of Chloroquine and Primaquine Linked by Gold(I): Multitarget and Multiphase Antiplasmodial Agent”, ChemMedChem, 16, 662-678
65. 117. D. Moita, H. Nunes-Cabaço, A.M. Mendes, M. Prudêncio (2021) “A guide to investigating immune responses elicited by whole-sporozoite pre-erythrocytic vaccines against malaria”, FEBS J., doi:10.1111/febs.16016
64. T.A. Tavella, N.S.M. Silva, N. Spillman, A.C.A.V.K., G.C. Cassiano, A.A. Vasconcelos, A.P. Camargo, D.C.B. Silva, D. Fontinha, L.C.S. Alvarez, L.T. Ferreira, K.C.P. Tomaz, B.J. Neves, L.D. Almeida, D.Y. Bargieri, M.V.G. Lacerda, P.V.L. Cravo, P. Sunnerhagen, M. Prudêncio, C.H. Andrade, S.C.P. Lopes, M.F. Carazzolle, L. Tilley, E. Bilsland, J.C. Borges, F.T.M. Costa (2021) “Violacein-Induced Chaperone System Collapse Underlies Multistage Antiplasmodial Activity” ACS Infect. Dis., 7, 759-776
63. N.G. Alves, I. Bártolo, A.J.S. Alves, D. Fontinha, D. Francisco, S.M.M. Lopes, M.I.L. Soares, C. J.V. Simões, M. Prudêncio, N. Taveira, T.M.V.D. Pinho e Melo (2021) “Synthesis and structure-activity relationships of new chiral spiro-b-lactams highly active against HIV-1 and Plasmodium”, Eur. J. Med. Chem., 219, 113439
62. M. Prudêncio (2021) “Portugal’s prominence in malaria research”, EMBO Reports, e51692
61. I Bártolo, B.S. Santos, D. Fontinha, M. Machado, D. Francisco, B. Sepodes, J. Rocha, H. Mota-Filipe, R. Pinto, M.E. Figueira, H. Barroso, T. Nascimento, A.P.A. de Matos, A.J.S. Alves, N.G. Alves, C.J.V. Simões, M. Prudêncio, T.M.V.D. Pinho e Melo, N. Taveira (2021) “Spiro-β-lactam BSS-730A displays potent activity against HIV and Plasmodium”, ACS Infectious Diseases, 7, 2, 421-434
60. M. Fonte, N. Tassi, D. Fontinha, I. Bouzón-Arnáiz, R. Ferraz, M.J. Araújo, X. Fernàndez-Busquets, M. Prudêncio, P. Gomes, C. Teixeira (2020) “4,9-diaminoacridines and 4-aminoacridines as antiplasmodial hits”. ChemMedChem, 16, 799-792
59. Y. Miyazaki, C.Y. Marin, T. Imai, A.M. Mendes, R. vd Laak, A. Sturm, F.J. Geurten, S. Miyazaki, S.C. Chevalley-Maurel, J. Ramesar, S.K. Kolli, J. Kroeze, R. van Schuijlenburg, A.M. Salman, B.K. Wilder, A. Reyes-Sandoval, K. Dechering, M. Prudêncio, C.J. Janse, S.M. Khan, B. Franke-Fayard (2020) “Generation of a genetically modified chimeric Plasmodium falciparum parasite expressing P. vivax circumsporozoite protein for malaria vaccine development”, Frontiers in Cellular and Infection Microbiology, 10, 591046
58. P. Meireles, D. Brás, D. Fontinha, A.F. Chora, K. Serre, A.M. Mendes*, M. Prudêncio* (2020) “Elimination of Hepatic Rodent Plasmodium Parasites by Amino Acid Supplementation”, iScience, 23, 101781 (*Corresponding authors). Recommended by Faculty Opinions
57. M. Marinović, I. Perković, D. Fontinha, M. Prudêncio, J. Held, L. Pessanha de Carvalho, T. Tandarić, R. Vianello, B. Zorc, Z. Rajić (2020) “Novel Harmicines with Improved Potency against Plasmodium”, Molecules, 25, 4376
56. M. Prudêncio (2020) "In fairness to mosquitoes", Trends in Parasitology, 36, 876-877
55. S.A. Milheiro, J. Gonçalves, R.M.R.M. Lopes, M. Madureira, L. Lobo, A. Lopes, F. Nogueira, D. Fontinha, M. Prudêncio, M.F.M. Piedade, S.N. Pinto, P.R. Florindo, R. Moreira (2020) “Half- sandwich cyclopentadienylruthenium(II) complexes: a new antimalarial chemotype”, Inorganic Chemistry, 59, 12722-12732
54. D. Fontinha, I. Moules, M. Prudêncio (2020) "Repurposing drugs to fight hepatic malaria parasites", Molecules, 25, 3409
53. M. Prudêncio, J.C. Costa (2020) "Research funding after COVID-19", Nature Microbiol., 5, 986
52. D. Fontinha, S.A. Sousa,
T.S. Morais, M. Prudêncio, J.H. Leitão, Y.L. Gal, D. Lorcy, R.A.L. Silva,
M.F.G. Velho, D. Belo, M. Almeida, J.F. Guerreiro, T. Pinheiro, F. Marques
(2020) "Gold(III) bis(dithiolene) complexes: from molecular conductors to
prospective anticancer, antimicrobial and antiplasmodial agents", Metallomics, 12, 974-987
51. I.J. Reuling *, A.M. Mendes*, G.M. de Jong GM*, A. Fabra-García*, H. Nunes-Cabaço*, G.J. van Gemert, W. Graumans, L.E. Coffeng, S.J. de Vlas, A.S.P. Yang, C.K. Lee, Y. Wu, A.J. Birkett, C.F. Ockenhouse, R. Koelewijn, J.J. van Hellemond, P.J.J. van Genderen**, R.W. Sauerwein**, M. Prudêncio** (2020) “Safety and efficacy of a genetically modified rodent malaria parasite against Plasmodium falciparum malaria: an open-label randomized phase 1/2a trial”, Science Transl. Med., 12, eaay2578. *Equally contributing authors; **Corresponding authors. Issue cover.
50. L. Singh, D. Fontinha, D. Francisco, A.M. Mendes, M. Prudêncio, K. Singh (2020) “Molecular Design and Synthesis of Ivermectin Hybrids Targeting Hepatic and Erythrocytic Stages of Plasmodium Parasites”, J. Med. Chem., 63, 1750-1762
49. R. Azevedo, A.M. Mendes, M. Prudêncio (2020) "The impact of antiretroviral therapy on malaria parasite transmission”, Frontiers in Microbiology-Infectious Diseases, 10, 3048
48. L. Balasubramanian, V. Zuzarte-Luís, T. Syed, D. Mullick, S. Deb, H. Prasad, J. Meissner, A.S. Almeida, T. Furstenhaupt, K. Siddiqi, M. Prudêncio, C.M. Rodrigues, M.M. Mota, V. Sundaramurthy (2020) "Association of Plasmodium berghei with the apical domain of hepatocytes is necessary for the parasite's liver stage development", Frontiers in Cellular Infection Microbiology, 9, 451
47. I. Perković, S. Raić-Malić, D. Fontinha, M. Prudêncio, L.P. Carvalho, J. Held, T. Tandarić, R. Vianello, B. Zorc, Zrinka Rajić (2020) "Harmicines − harmine and cinnamic acid hybrids as novel antiplasmodial hits", Eur. J. Med. Chem., 187, 111927
46. S.A. Sousa, J.H. Leitão, R.A.L. Silva, D. Belo, I.C. Santos, J.F. Guerreiro, M. Martins, D. Fontinha, M. Prudêncio, M. Almeida, D. Lorcy, F. Marques (2020) "On the Path to Gold: Monoanionic Au Bisdithiolate Complexes with 1 Antimicrobial and Antitumor Activities", Journal of Inorganic Biochemistry, 202, 110904
45. A.J.S. Alves, N.G. Alves, C.C. Caratão, Esteves M., D. Fontinha, I. Bártolo, M.I.L. Soares, S.M.M. Lopes, M. Prudêncio, N. Taveira, T.M.V.D. Pinho e Melo (2019) "Spiro-Lactams as Novel Antimicrobial Agents", Curr. Top. Med. Chem., 20, 140-152
44. M. Sanches-Vaz, A. Temporão, R. Luis, H. Nunes-Cabaço, A.M. Mendes, S. Goellner, T. Carvalho, L.M. Figueiredo*, M. Prudêncio* (2019) "Trypanosoma brucei infection protects mice against malaria", PLoS Pathogens, 15, e1008145 (* Corresponding authors)
43. R. Azevedo, A.M. Mendes, M.Prudêncio (2019) "Inhibition of Plasmodium sporogonic stages by ivermectin and other avermectins", Parasites & Vectors, 12, 594
42. F. Arez, S. Rebelo, D. Fontinha, D. Simão, T.R. Martins, M. Machado, C. Fischli, C. Oeuvray, L. Badolo, M. J. T. Carrondo, M. Rottmann, T. Spangenberg, C. Brito, B. Greco*, M. Prudêncio*, P.M. Alves* (2019) “Flexible 3D cell-based platforms for the discovery and profiling of novel drugs targeting Plasmodium hepatic infection”, ACS Infect. Dis., 5, 1831-1842 (* Corresponding authors)
36. G. Mayoka, M. Njoroge, J. Okombo, L.
Gibhard, M. Sanches-Vaz, D. Fontinha, L.M. Birkholtz, J. Reader, M. van der
Watt, T.L. Coetzer, S. Lauterbach, A. Churchyard, B. Bezuidenhout, T.J. Egan,
C.L. Yeates, S. Wittlin, M. Prudêncio, K. Chibale (2019) “Structure-activity
relationship studies and Plasmodium life cycle profiling identifies pan-active
N-aryl-3-trifluoromethyl pyrido[1,2-a]benzimidazoles which are efficacious in
an in vivo mouse model of malaria”, J. Med. Chem., 62, 1022-1035
35. M. Kumar, J. Okombo, D. Mambwe, D. Taylor, N. Lawrence, J. Reader, M.V. Watt, D. Fontinha, M. Sanches-Vaz, B. Bezuidenhout, S. Lauterbach, D. Liebenberg, L.M. Birkholtz, T.L. Coetzer, M. Prudêncio, T.J. Egan, S. Wittlin, K. Chibale (2019) “Multistage Antiplasmodium Activity of Astemizole Analogues and Inhibition of Hemozoin Formation as a Contributor to Their Mode of Action”, ACS Infect. Dis., 5, 303-315
32. A.M. Mendes, M. Machado, N. Gonçalves-Rosa, I.J. Reuling, L. Foquet, C. Marques, A.M. Salman, A.S.P. Yang, K.A. Moser, A. Dwivedi, C.C. Hermsen, B. Jiménez-Díaz, S. Viera, J.M. Santos, I. Albuquerque, S.N. Bhatia, J. Bial, I. Angulo-Barturen, J.C. Silva, G. Leroux-Roels, C.J. Janse, S.M. Khan, M.M. Mota, R.W. Sauerwein, M. Prudêncio (2018) "A Plasmodium berghei Sporozoite-Based Vaccination Platform Against Human Malaria", NPJ Vaccines, 3, 33
30. M. Šafratová, A. Hošťálková, D. Hulcová, K. Breiterová, V. Hrabcová, M. Machado, D. Fontinha, M. Prudêncio, J. Kuneš, J. Chlebek, D. Jun, M. Hrabinová, L. Nováková, R. Havelek, M. Seifrtová, L. Opletal, L. Cahlíková (2018) "Alkaloids from Narcissus poeticus cv. Pink Parasol of various structural types and their biological activity", Arch. Pharmacal Res., 41, 208-218
29. K. Pavic, I. Perkovic, S. Popisilova, M. Machado, D. Fontinha, M. Prudêncio, J. Jampilek, A. Coffey, L. Endersen, H. Rimac, B. Zorc (2017) "Primaquine hybrids as promising antimycobacterial and antimalarial agents", Eur. J. Med. Chem., 143, 769-779
28. T.S. Macedo, W. Villarreal, C.C. Couto, D.R.M. Moreira, M. Navarro, M. Machado, M. Prudêncio, A.A. Batista, M.B.P. Soares (2017) "Platinum(II)-chloroquine complexes are antimalarial agents against blood and liver stages by impairing mitochondrial function", Metallomics, 9, 1548-1561
27. M. Machado, M. Sanches-Vaz, J.P. Cruz, A.M. Mendes, M. Prudêncio (2017) "Inhibition of Plasmodium hepatic infection by antiretroviral compounds", Front. Cell. Infect. Microbiol., 7, doi: 10.3389/fcimb.2017.00329
26. P. Meireles, A.M. Mendes, R.I. Aroeira, B.C. Mounce, M. Vignuzzi, H.M. Staines, M. Prudêncio (2017) "Uptake and metabolism of arginine impact Plasmodium development in the liver", Sci. Rep., 7, 4072
25. R. Azevedo§, M. Markovic§, M. Machado, B. Franke-Fayard, A.M. Mendes*, M. Prudêncio* (2017) "A bioluminescence method for in vitro screening of Plasmodium transmission-blocking compounds", Antimicrob. Agents Chemother., 61, 202699-16. §- Equally contributing authors; *- Corresponding authors
24. K. Singh, J. Okombo, C. Brunschwig, F. Ndubi, L. Barnard, C. Wilkinson, P.M. Njogu, M. Njoroge, L. Laing, M. Machado, M. Prudêncio, J. Reader, M. Botha, S. Nondaba, L.M. Birkholtz, S. Lauterbach, A. Churchyard, T.L. Coetzer, J.N. Burrows, C. Yeates, P. Denti, L. Wiesner, T.J. Egan, S. Wittlin, K. Chibale (2017) "Antimalarial pyrido[1,2-a]benzimidazoles: Lead optimization, parasite life cycle stage profile, mechanistic evaluation, killing kinetics and in vivo oral efficacy in a mouse model", J. Med. Chem., 60, 1432-1448
23. C.S. Cunha§, B. Nyboer§, K. Heiss, M. Sanches-Vaz, D. Fontinha, E. Wiedtke, D. Grimm, J.M. Przyborski, M.M. Mota, M. Prudêncio*, A.K. Mueller* (2017) "P. berghei EXP-1 Interacts with Host Apolipoprotein H during Plasmodium Liver Stage Development", Proc. Natl. Acad. Sci. USA, 114, E1138-E1147. §- Equally contributing authors; *- Corresponding authors
22. A.M. Mendes, I.S. Albuquerque, M. Machado, J. Pissarra, P. Meireles, M. Prudêncio (2017) "Inhibition of Plasmodium liver infection by ivermectin", Antimicrob. Agents Chemother., 61, e02005-16
21. M.A.S. Cavadas, M.P. Monopoli, C.S. Cunha, M. Prudêncio, E. Pereira, I. Lynch, K.A. Dawson, R. Franco (2016) "Unravelling Malaria Antigen Binding to Antibody-Gold Nanoparticle Conjugates", Particle & Particle Systems Characterization, 33, 906-915
20. Carrasco M.P.*, Machado M., Gonçalves L., Sharma M., Gut J., Lukens A.K., Wirth D.F., André V., Duarte M.T., Guedes R.C., Dos Santos D., Rosenthal P.J., Mazitschek R., Prudêncio M.*, Moreira R. (2016) "Probing the Azaaurone Scaffold against the Hepatic and Erythrocytic Stages of Malaria Parasites", ChemMedChem, 11, 2194-2204 (* Corresponding authors)
19. P. Meireles, J. Sales-Dias, C.M. Andrade, J. Mello-Vieira, L. Mancio-Silva, J.P. Simas, H.M. Staines, M. Prudêncio (2016) "GLUT1-mediated glucose uptake plays a crucial role during Plasmodium hepatic infection", Cell. Microbiol., doi:10.1111/cmi.12646
18. R. Ferraz, J. Noronha, F. Murtinheira, F. Nogueira, M. Machado, M. PrudêncioB., S. Parapini, S. D’Alessandro, C. Teixeira, A. Gomes, C. Prudêncio, P. Gomes (2016) "Primaquine-based ionic liquids as a novel class of antimalarial hits", RSC Advances, 6, 56134-56138
17. T.S. Macedo, L.C. Vegas, M. Paixão, M. Navarro, B.C. Barreto, P.C.M..Oliveira, S.G. Macambira, M. Machado, M. Prudêncio, S. D’Alessandro, N. Basilico, D.R.M. Moreira, A.A. Batista, M.B.P. Soares (2016) "Chloroquine-containing organoruthenium complexes are fast-acting multistage antimalarial agents", Parasitology, 143, 1543-1556
16. C.J.A. Ribeiro, M. Espadinha, M. Machado, J. Gut, L.M. Gonçalves, P.J. Rosenthal, M. Prudêncio, R. Moreira, M.M.M. Santos (2016) "Novel squaramides with in vitro liver stage antiplasmodial activity", Bioorg. Med. Chem., 24, 1786-1792
15. N. Terzić, J. Konstantinović, M. Tot, J. Burojević, O. Djurković-Djaković, J. Srbljanović, T. Štajner, T. Verbić, M. Zlatović, M. Machado, I.S. Albuquerque, M. Prudêncio*, R.J. Sciotti, S. Pecic, S. D’Alessandro, D. Taramelli, B.A. Šolaja* (2016) "Re-investigating old pharmacophores: Are 4-aminoquinolines and tetraoxanes potential two-stage antimalarials?", J. Med. Chem., 59, 264-281 (* Corresponding authors)
14. I. Gomes, A. Reis, E. Pereira, E. Fortunato, M. Prudêncio, R. Franco (2015) "Nanoimunoensaios para diagnóstico de malária", An. Inst. Hig. Med. Trop., 14, 21-30
13. N.A.L. Pereira, Â. Monteiro, M. Machado, J. Gut, E. Molins, M.J. Perry, J. Dourado, R. Moreira, P.J. Rosenthal, M. Prudêncio*, and M.M.M. Santos* (2015), "Enantiopure Indolizinoindolones with in vitro Activity against Blood- and Liver-Stage Malaria Parasites". ChemMedChem, 10, 2080-2089 (* Corresponding authors)
12. A. Gomes, M. Machado, L. Lobo, F. Nogueira, M. Prudêncio, C. Teixeira, P. Gomes (2015) "N-cinnamoylation of antimalarial classics: Effects of using acyl groups other than cinnamoyl toward dual-stage antimalarials", ChemMedChem, 10, 1344-134
11. H. Kaur, M. Machado, C. de Kock, P. Smith, K Chibale, M Prudêncio, K. Singh (2015) "Primaquineepyrimidine hybrids: Synthesis and dual-stage antiplasmodial activity", European Journal of Medicinal Chemistry, 101, 266-273
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